Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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Thermo Scientific Chemicals Olaparib
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Thermo Scientific Chemicals Olaparib
CAS: 763113-22-0 Molecular Formula: C24H23FN4O3
| CAS | 763113-22-0 |
|---|---|
| Molecular Formula | C24H23FN4O3 |
64
R&D Systems™ Cy5-Fuc Labeled N2f
Small and Specialty Supplier Partner
Small and/or specialty supplier based on Federal laws and SBA requirements.
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65
Tocris Bioscience™ CRT 0105950
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent LIMK1/2 inhibitor
66
Tocris Bioscience™ Ivacaftor
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective CFTR potentiator
| Target | CFTR |
|---|---|
| CAS | 873054-44-5 |
| Purity | 98% |
| Chemical Name or Material | N-[2,4-Bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxo-3-quinolinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H28N2O3 |
67
Tocris Bioscience™ AP 14145 hydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Negative allosteric modulator of KCa2 (SK) channels
68
Tocris Bioscience™ LW 6
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Malate dehydrogenase-2 (MDH2) inhibitor; also inhibits HIF-1α
| Target | Dehydrogenase Inhibitors |
|---|---|
| CAS | 934593-90-5 |
| Purity | 0.98 |
| Chemical Name or Material | Methyl 4-hydroxy-3-[[2-(4-tricyclo[3.3.1.13,7 ]dec-1-ylphenoxy)acetyl]amino]benzoate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C26H29NO5 |
69
Tocris Bioscience™ ent-LP 99
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Negative Control for LP 99
| CAS | 1808948-28-8 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[(2S,3R)-2-(4-Chlorophenyl)-1-(1,2-dihydro-1,4-dimethyl-2-oxo-7-quinolinyl)-6-oxo-3-piperidinyl]-2-methyl-1-propanesulfonamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C26H30ClN3O4S |
| Formula Weight | 516.05 |
70
Tocris Bioscience™ Squarunkin A Hydrochloride
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UNC119 chaperone-cargo interaction inhibitor; disrupts Src activation
| Purity | 98% |
|---|---|
| Chemical Name or Material | Ethyl 4-((3,4-dioxo-2-((2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)amino)cyclobut-1-en-1-yl)amino)piperidine-1-carboxylate hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H32F3N5O4.HCl |
| Formula Weight | 560.01 |
71
Tocris Bioscience™ PARPi-FL
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Small and Specialty Supplier Partner
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Potent fluorescent PARP inhibitor
72
Tocris Bioscience™ SU 6656
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Potent ATP-competitive Src family kinase inhibitor (IC50 values are 0.02, 0.13, 0.17, 0.28 and 6.88 nM for Yes, Lyn, Fyn, Src and Lck, respectively)
| CAS | 330161-87-0 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 2,3-Dihydro-N,N-dimethyl-2-oxo-3-[(4,5,6,7-tetrahydro-1H-indol-2-yl)methylene]-1H-indole-5-sulfonamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H21N3O3S |
| Formula Weight | 371.45 |
73
Tocris Bioscience™ EM12-SO2F
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent covalent inhibitor of Cereblon
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Thermo Scientific Chemicals Tiotropium bromide
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Thermo Scientific Chemicals Tiotropium bromide
CAS: 139404-48-1 Molecular Formula: C19H22BrNO4S2
| CAS | 139404-48-1 |
|---|---|
| Molecular Formula | C19H22BrNO4S2 |
75
Tocris Bioscience™ CU CPT 9a
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Potent TLR8 inhibitor
| CAS | 2165340-32-7 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 2-Methyl-4-(7-methoxy-4-quinolinyl)phenol |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C17H15NO2 |