Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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61
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75
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60,533
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61
R&D Systems™ MK 2206 dihydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective allosteric Akt1, Akt2 and Akt3 inhibitor
| Target | Akt (Protein Kinase B) Inhibitors |
|---|---|
| CAS | 1032350-13-2 |
| Purity | 0.98 |
| Chemical Name or Material | 8-[4-(1-Aminocyclobutyl)phenyl]-9-phenyl-1,2,4-triazolo[3,4-f][1,6]naphthyridin-3(2H)-one dihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H21N5O.2HCl |
62
| CAS | 19685-09-7 |
|---|---|
| Molecular Formula | C20H16N2O5 |
63
R&D Systems™ MR 24
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective MST3 kinase binding inhibitor
| Target | Other Kinase Inhibitors |
|---|---|
| Purity | 0.98 |
| Chemical Name or Material | 8-(4-Aminobutyl)-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(1,3-dihydroxypropan-2-ylamino)pyrido[2,3-d]pyrimidin-7-one trihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C26H29ClN6O3.3HCl |
64
R&D Systems™ Thalidomide 4'-oxyacetamide-alkylC8-amine
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with alkyl linker and terminal amine for onward chemistry
65
R&D Systems™ Lapatinib
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective dual ErbB2 (HER-2) and EGFR inhibitor (IC50 values are 9.8 and 10.2 nM, respectively)
| CAS | 231277-92-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C29H26ClFN4O4S |
| Formula Weight | 581.06 |
66
R&D Systems™ Conivaptan Hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Very high affinity vasopressin V1A and V2 antagonist; orally bioavailable
| CAS | 168626-94-6 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[4-[(4,5-Dihydro-2-methylimidazo[4,5-d][benzazepin-6(1H)-yl)carbonyl]phenyl-[1,1'-biphenyl]-2-carboxamide hydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C32H26N4O2.HCl |
| Formula Weight | 535.04 |
67
Thermo Scientific Chemicals Ligustrazine hydrochloride
CAS: 76494-51-4 Molecular Formula: C8H12N2·HCl
| CAS | 76494-51-4 |
|---|---|
| Molecular Formula | C8H12N2·HCl |
68
| CAS | 55079-83-9 |
|---|---|
| Molecular Formula | C21H26O3 |
69
R&D Systems™ Ortho AP 1867
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Selective binding ligand for FKBP12F36V; precursor for dTAG compounds
| Target | FKBP12 |
|---|---|
| CAS | 2230613-03-1 |
| Purity | 0.98 |
| Chemical Name or Material | 2-(2-((R)-3-(3,4-Dimethoxyphenyl)-1-(((S)-1-((S)-2-(3,4,5-trimethoxyphenyl)butanoyl)piperidine-2-carbonyl)oxy)propyl)phenoxy)acetic acid |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C38H47NO11 |
70
| CAS | 53902-12-8 |
|---|---|
| Color | White to Light-yellow to Green |
| Solubility | insoluble in water |
| Physical Form | Crystalline Powder |
| Health Hazard 1 | GHS07: Exclamation mark |
| Chemical Name or Material | Tranilast |
| Recommended Storage | Refrigerator +4°C |
| Merck Index | 9646 |
| Molecular Formula | C18 H17 N O5 |
| Formula Weight | 327.33 |
| Melting Point | 166.2°C to 168.2°C |
71
R&D Systems™ GSK 626616
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective DYRK inhibitor; orally bioavailable.
| CAS | 1025821-33-3 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (5Z)-2-[(2,6-Dichlorophenyl)amino]-5-(6-quinoxalinylmethylene)-4(5H)-thiazolone |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C18H10Cl2N4OS |
| Formula Weight | 401.27 |
73
R&D Systems™ BI 3231
A Tocris product, part of R&D Systems. Potent and selective hydroxysteroid 17β dehydrogenase 13 (HSD17B13) inhibitor
74
R&D Systems™ AZ 5704
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective ATM kinase inhibitor; orally bioavailable
| CAS | 1941214-06-7 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 7-Fluoro-6-[6-(methoxymethyl)-3-pyridinyl]-4-[[(1S)-1-(1-methyl-1H-pyrazol-3-yl)ethyl]amino]-3-quinolinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H23FN6O2 |
| Formula Weight | 434.47 |
75
R&D Systems™ Thalidomide 4'-ether-alkylC6-amine
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Thalidomide-alkylC6-amine